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Humanin

A compound studied for protecting the brain and keeping cells alive and insulin-sensitive as you age. A mitochondrial-derived peptide encoded inside mitochondrial DNA, studied for neuroprotection, insulin sensitivity, and cellular survival.

Longevity
Evidence: Limited

Humanin: A compound studied for protecting the brain and keeping cells alive and insulin-sensitive as you age. A mitochondrial-derived peptide encoded inside mitochondrial DNA, studied for neuroprotection, insulin sensitivity, and cellular survival. Humanin is a peptide your mitochondria make and secrete.

FDA
Not approved
WADA
Not banned
Typical dose
1-10 mg sub-q daily
Half-life
~minutes (rapid clearance)
Route
Subcutaneous
Schedule
Daily
In plain English

Humanin is a peptide your mitochondria make and secrete. It's tied to neuroprotection, insulin sensitivity, and cellular survival. Slow, subtle effects, mostly used as a longevity-stack add-on.

Status & legalityWhat do these mean? →
Natty?
Grey area

Mitochondrial-derived peptide. Naturally produced; exogenous use is a different question.

FDA
Not approved

Not FDA approved.

Compounding
Not classified

Not formally categorized in the FDA bulks lists.

WADA
Not listed
Prescribed

Not prescribed in conventional medicine.

Who it's for

  • Users running longevity-focused stacks
  • Older adults targeting metabolic and neuroprotective markers
  • Cellular bioenergetics enthusiasts

What to expect

  1. Week 1

    Subtle. Energy and mood lift first for responders.

  2. Week 4

    Cumulative metabolic / cognitive support.

  3. Week 8

    Plateau. Cycle off.

Looking at Humanin? Your next 3 steps

  1. 1Work out your syringe units

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  2. 2See what to stack & monitor

    The companion supplements and the bloodwork worth tracking on this kind of protocol.

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  3. 3Save it & ask the Coach

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How it works (mechanism)

Mitochondrial-derived peptide encoded inside mitochondrial DNA. Binds receptors that activate STAT3 and reduce apoptosis, particularly in neurons and pancreatic beta cells.

Dosing protocol

Members only

Stacks well with

Members only

Side effects

01Generally well tolerated
02Limited safety data, short cycles preferred

When NOT to use

  • Pregnancy / nursing
  • No data in active malignancy

Bloodwork to monitor

  • Fasting glucose / insulin if running longer

Common mistakes

  • Expecting fast or visible effects (it's slow and subtle)
  • Stacking with too many longevity peptides simultaneously
  • Running indefinitely, limited human safety data

What it actually is

Humanin is a small peptide encoded within mitochondrial DNA, with nuclear-encoded humanin-like sequences also described — one of the same small family as MOTS-c. It was discovered in 2001 in the brain tissue of an Alzheimer's patient, in the region that had survived, which is where its neuroprotective reputation comes from. It has never been approved and there are nine indexed human-trial records, none establishing a clinical outcome.

Humanin appears to act as a cellular survival signal. It interferes with apoptosis — programmed cell death — by binding pro-apoptotic proteins, and it acts on a cell-surface receptor complex to trigger protective signalling. Circulating levels have been reported to fall with age and to be higher in the children of long-lived parents, though the human data on the age association is inconsistent. That is the basis for the longevity interest. That is an association in observational data, not a demonstration that raising it does anything.

Forms, and which is which

Lyophilised powder, subcutaneousHow all use happens

Buyer reconstitutes. Research-chemical supply with unverified identity, at doses extrapolated from animal work.

Verdict: The only form, unregulated.

Humanin analogs (HNG and others)Research potency

Modified versions used in research because they are far more potent than the native peptide. What is sold is rarely specified as either.

Verdict: Ask which one; the answer is usually unavailable.

MOTS-c and other mitochondrial peptidesThe same family

Same class of mitochondrially encoded peptides, different proposed actions.

Verdict: Related biology, separately unproven.

Oral preparationsNothing

Not absorbed intact as an active dose.

Verdict: Not plausible by the route claimed.

What it is claimed to do, graded

Protects neurons from amyloid toxicityLimited

The founding observation, demonstrated in cell and animal models of Alzheimer's disease over two decades. Genuinely interesting, entirely preclinical.

Improves insulin sensitivityLimited

Shown in animal models. No human trial.

Higher levels associate with longevityLimited

Observational: levels fall with age and are higher in offspring of long-lived people. Association, and one that does not establish direction of causation.

Extends lifespan or slows ageing in humansNone shown

No human data of any kind.

Protects against neurodegeneration in peopleNone shown

The reason most people take it. Cell and animal models only.

Grades describe how much human evidence exists for that specific claim, not whether it will work for you or whether it is safe.

Pros and cons

Pros
  • Genuinely novel biology — a mitochondrially encoded peptide is a real discovery
  • A substantial preclinical literature spanning two decades
  • The Alzheimer's origin story is real, not marketing
  • No serious harms reported, on no human administration data — absence of reports rather than a safety finding
Cons
  • Nine indexed human records, which observe endogenous humanin rather than test giving it, and none establishing a clinical outcome
  • Very short half-life, so how any injected dose produces a sustained effect is unclear
  • The longevity association is observational and could run either direction
  • Anti-apoptotic activity is exactly what you do not want near a cell that should be dying
  • Research-chemical supply with unverified identity

When to stop

  • Any new lump or unexplained weight loss
  • You are undergoing or about to start cancer treatment
  • Injection-site reaction that spreads
  • You are running it continuously with nothing to measure

Interactions

Active or suspected cancerAvoid

Humanin suppresses apoptosis. Preventing damaged cells from dying is the mechanism you least want near a tumour, and this is a real rather than pro-forma concern.

ChemotherapyAvoid

Many chemotherapy agents work by triggering apoptosis, so an anti-apoptotic signal would be expected to oppose them. Predicted from mechanism rather than demonstrated, and not a risk worth taking during treatment.

Other mitochondrial peptidesCaution

Stacking compounds without human evidence makes any effect unattributable.

Diabetes medicationMonitor

If the insulin-sensitivity effect is real it works in the same direction.

Nothing well characterisedCaution

There is no human interaction literature for this compound.

Is this for you?

Probably worth reading further if
  • People who find the mitochondrial-peptide biology interesting and accept they are well ahead of the evidence
Skip it if
  • You have active cancer or any undiagnosed lump — the anti-apoptotic mechanism is the specific concern
  • You are undergoing chemotherapy
  • You are pregnant or nursing
  • You want a measurable result — there is nothing here you can check

The one number

9 indexed human-trial records and zero establishing a clinical outcome
Pepdex evidence index — counts are indexed PubMed records, not deduplicated trials; PubMed query for humanin

Sources for the claims above

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AI Coach, live sample
Member answer
is 250mcg of bpc enough for a knee injury?
For a knee, is the standard working dose and a solid place to start. The trick with BPC is consistency, give it weeks, not days. , run it , and don't drop below , results tend to fall off under that line. If nothing's moved by week 3, that's when earns its place.
how much bac water for a 10mg reta vial?
is the standard play for a 10 mg reta vial. That gives you , clean unit math across the whole titration: on a 100-unit insulin syringe. Run instead if you want fewer, more concentrated shots. Most people titrate up over , and that mix keeps the numbers cleanest.
what should i track on bloodwork for tirzepatide?
Lipid panel, ALT/AST (liver enzymes), and an A1C, baseline before you start then every 3 months. If you've got metabolic-syndrome history, add fasting glucose and insulin so you can actually watch insulin sensitivity improve. You don't need a big hormone panel for a GLP-1.

Numbers redacted in this preview. Members get the full answer, on their own stack.

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Frequently asked

What is Humanin?+
Humanin is a peptide your mitochondria make and secrete. It's tied to neuroprotection, insulin sensitivity, and cellular survival. Slow, subtle effects, mostly used as a longevity-stack add-on.
Is Humanin FDA approved?+
Not FDA approved.
Is Humanin legal?+
Humanin is not FDA-approved, so there is no approved prescription version. Most supply is sold as "research only" by peptide vendors. A compounding pharmacy may only use substances the FDA permits for compounding, and many research peptides are not permitted — do not assume a compounded prescription is available. Possession is generally not criminalized but distribution without authorization may be. Verify local laws.
Is Humanin banned by WADA?+
Humanin is not currently on the WADA prohibited list.
Are you still natty after taking Humanin?+
Grey area. Mitochondrial-derived peptide. Naturally produced; exogenous use is a different question.
Do doctors prescribe Humanin?+
Not prescribed in conventional medicine.
What's the typical dose of Humanin?+
Dosing depends on your goal, experience, and tolerance. The full Humanin protocol (dose, frequency, and how to titrate) is in the members section on the entry page.
What are the side effects of Humanin?+
Common side effects include: Generally well tolerated; Limited safety data, short cycles preferred. Less common effects and full safety details are on the entry page.
How long until Humanin starts working?+
Subtle. Energy and mood lift first for responders.
What can you stack with Humanin?+
Humanin is commonly combined with complementary compounds. The full stacking protocol (what to pair, dosing, and timing) is in the members section on the entry page.
Where do people get Humanin?+
Pepdex does not sell, ship, or recommend suppliers. Humanin is not FDA-approved; prescription versions require licensed clinical care, and "research only" markets carry real legal and quality risks. /coa explains how to verify a Certificate of Analysis and /guides/scam-vendor-spotting covers the red flags.

Common questions about Humanin